YASUHARA, Akito: search on Z-Library

The world's largest scientific articles store. 70,000,000+ articles for free.

1

Identification of 1-Methyl-N-(propan-2-yl)-N-({2-[4-(trifluoromethoxy)phenyl]pyridin-4-yl}methyl)-1H-imidazole-4-carboxamide as a Potent and Orally Available Glycine Transporter 1 Inhibitor

Yamamoto, Shuji, Ohta, Hiroshi, Abe, Kumi, Kambe, Daiji, Tsukiyama, Naohiro, Kawakita, Yasunori, Moriya, Minoru, Yasuhara, Akito

Year:

2016

Language:

english

File:

PDF, 1.10 MB

english, 2016

2

Condensed heteroaromatic ring systems. XVIII. Palladium-catalyzed cross-coupling reaction of aryl bromides with (Z)-1-ethoxy-2-tributylstannylethene and its utilization for construction of condensed heteroaromatics

Takao Sakamoto, Yoshinori Kondo, Akito Yasuhara, Hiroshi Yamanaka

Journal:

Year:

1991

Language:

english

File:

PDF, 632 KB

english, 1991

3

Selective Monodesulfonylation of N,N-Disulfonylarylamines with Tetrabutylammonium Fluoride.

YASUHARA, Akito, KAMEDA, Mitsuyoshi, SAKAMOTO, Takao

Journal:

CHEMICAL & PHARMACEUTICAL BULLETIN

Year:

1999

File:

PDF, 771 KB

1999

4

Total syntheses of three natural products, vignafuran, 2-(4-hydroxy-2-methoxyphenyl)-6-methoxybenzofuran-3-carboxylic acid methyl ester, and coumestrol from a common starting material

Hiroya, Kou, Suzuki, Naoyuki, Yasuhara, Akito, Egawa, Yuya, Kasano, Atsushi, Sakamoto, Takao

Journal:

Journal of the Chemical Society Perkin Transactions 1

Year:

2000

Language:

english

File:

PDF, 249 KB

english, 2000

5

ChemInform Abstract: Total Syntheses of Three Natural Products, Vignafuran, 2-(4-Hydroxy-2-methoxyphenyl)-6-methoxybenzofuran-3-carboxylic Acid Methyl Ester, and Coumestrol from a Common Starting Material.

Kou Hiroya, Naoyuki Suzuki, Akito Yasuhara, Yuya Egawa, Atsushi Kasano, Takao Sakamoto

Journal:

Year:

2001

File:

PDF, 31 KB

2001

6

Cyclization reactions of 2-alkynylbenzyl alcohol and 2-alkynylbenzylamine derivatives promoted by tetrabutylammonium fluoride

Kou Hiroya, Rumi Jouka, Mitsuyoshi Kameda, Akito Yasuhara, Takao Sakamoto

Journal:

Year:

2001

Language:

english

File:

PDF, 276 KB

english, 2001

7

Contrasting fates for 6-α-methylpenicillin N upon oxidation by deacetoxycephalosporin C synthase (DAOCS) and deacetoxy/deacetylcephalosporin C synthase (DAOC/DACS)

Christopher S Hamilton, Akito Yasuhara, Jack E Baldwin, Matthew D Lloyd, Peter J Rutledge

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 171 KB

english, 2001

8

ChemInform Abstract: A Concise Synthesis of Furostifoline by Tetrabutylammonium Fluoride-Promoted Indole Ring Formation.

Akito Yasuhara, Naoyuki Suzuki, Takao Sakamoto

Journal:

Year:

2002

File:

PDF, 28 KB

2002

9

ChemInform Abstract: Convenient Reduction of Nitrobenzenes to Anilines Using Electrochemically Generated Nickel.

Akito Yasuhara, Atsushi Kasano, Takao Sakamoto

Journal:

Year:

1999

File:

PDF, 36 KB

1999

10

Synthesis of Ethoxyethynylarenes by the Palladium-Catalyzed Reaction of Aryl Iodides with Ethoxy(trialkylstannyl)acetylenes.

SAKAMOTO, Takao, YASUHARA, Akito, KONDO, Yoshinori, YAMANAKA, Hiroshi

Journal:

CHEMICAL & PHARMACEUTICAL BULLETIN

Year:

1994

File:

PDF, 707 KB

1994

11

Pancreastatin-like immunoreactivity in globular dystrophic neurites of senile plaques in brains of patients with Alzheimer's disease

Osamu Yasuhara, Ichiro Akiguchi, Shinichi Nakamura, Ayae Kinoshita, Akito Ikemoto, Yasuhiro Kawamoto, Jun Kimura, Akihiro Funakoshi, Kayoko Tateishi, Patrick L. McGeer

Journal:

Neuroscience Letters

Year:

1996

Language:

english

File:

PDF, 838 KB

english, 1996

12

An Efficient Method for the Deallylation of Allyl Aryl Ethers Using Electrochemically Generated Nickel

Yasuhara, Akito, Kasano, Atsushi, Sakamoto, Takao

Journal:

Journal of Organic Chemistry

Year:

1999

Language:

english

File:

PDF, 77 KB

english, 1999

13

Antipsychotic profiles of TASP0443294, a novel and orally active positive allosteric modulator of metabotropic glutamate 2 receptor

Hikichi, Hirohiko, Hiyoshi, Tetsuaki, Marumo, Toshiyuki, Tomishima, Yasumitsu, Kaku, Ayaka, Iida, Izumi, Urabe, Hiroki, Tamita, Tomoko, Yasuhara, Akito, Karasawa, Jun-ichi, Chaki, Shigeyuki

Journal:

Journal of Pharmacological Sciences

Year:

2015

Language:

english

File:

PDF, 1.22 MB

english, 2015

14

Palladium-Catalyzed Cross-Coupling Reaction of Ethoxy(tributylstannyl)acetylene with Aryl Iodides

Sakamoto, Takao, Yasuhara, Akito, Kondo, Yoshinori, Yamanaka, Hiroshi

Journal:

Year:

1992

File:

PDF, 77 KB

1992

15

ChemInform Abstract: Electrochemical Generation of Highly Reactive Nickel and Its Utilization for Organic Reactions

Akito Yasuhara, Atsushi Kasano, Takao Sakamoto

Journal:

Year:

2000

File:

PDF, 25 KB

2000

16

Convenient indole synthesis from ethynylanilines with a polymer-supported fluoride

Akito Yasuhara, Naoyuki Suzuki, Takashi Yoshino, Yousuke Takeda, Takao Sakamoto

Journal:

Tetrahedron Letters

Year:

2002

Language:

english

File:

PDF, 70 KB

english, 2002

17

Novel synthetic strategy of carbolines via palladium-catalyzed amination and arylation reaction

Iwaki, Takehiko, Yasuhara, Akito, Sakamoto, Takao

Journal:

Journal of the Chemical Society Perkin Transactions 1

Year:

1999

Language:

english

File:

PDF, 154 KB

english, 1999

18

ChemInform Abstract: Synthesis of 2,3-Disubstituted Indole Using Palladium(II)-Catalyzed Cyclization with Alkenylation Reaction.

Akito Yasuhara, Yousuke Takeda, Naoyuki Suzuki, Takao Sakamoto

Journal:

Year:

2002

File:

PDF, 33 KB

2002

19

Synthesis, in vitro pharmacology, and structure–activity relationships of 2-aminobicyclo[3.1.0]hexane-2,6-dicarboxylic acid derivatives as mGluR2 antagonists

Akito Yasuhara, Kazunari Sakagami, Ryoko Yoshikawa, Shigeyuki Chaki, Masato Nakamura, Atsuro Nakazato

Journal:

Bioorganic & Medicinal Chemistry

Year:

2006

Language:

english

File:

PDF, 379 KB

english, 2006

20

Convenient synthesis of 2-substituted indoles from 2-ethynylanilines with tetrabutylammonium fluoride

Yasuhara, Akito, Kanamori, Yuichi, Kaneko, Masashi, Numata, Atsushi, Kondo, Yoshinori, Sakamoto, Takao

Journal:

Journal of the Chemical Society Perkin Transactions 1

Year:

1999

Language:

english

File:

PDF, 170 KB

english, 1999

21

ChemInform Abstract: An Efficient Method for the Deallylation of Allyl Aryl Ethers Using Electrochemically Generated Nickel.

Akito Yasuhara, Atsushi Kasano, Takao Sakamoto

Journal:

Year:

1999

File:

PDF, 31 KB

1999

22

Electrochemical Generation of Highly Reactive Nickel and Its Utilization for the Dehalogenative Coupling of Aryl Halides

Yasuhara, Akito, Kasano, Atsushi, Sakamoto, Takao

Journal:

Organometallics

Year:

1998

Language:

english

File:

PDF, 58 KB

english, 1998

23

ChemInform Abstract: Convenient Synthesis of 2-Substituted Indoles from 2-Ethynylanilines with Tetrabutylammonium Fluoride.

Akito Yasuhara, Yuichi Kanamori, Masashi Kaneko, Atsushi Numata, Yoshinori Kondo, Takao Sakamoto

Journal:

Year:

1999

File:

PDF, 28 KB

1999

24

Synthesis of 2-Substituted 3-Alkenyl-indoles by the Palladium-catalyzed Cyclization Followed by Alkenylation (Heck Reaction)

Sakamoto, Takao, Yasuhara, Akito, Kaneko, Masashi

Journal:

Year:

1998

Language:

english

File:

PDF, 190 KB

english, 1998

25

Convenient Reduction of Nitrobenzenes to Anilines Using Electrochemically Generated Nickel

Yasuhara, Akito, Kasano, Atsushi, Sakamoto, Takao

Journal:

Journal of Organic Chemistry

Year:

1999

Language:

english

File:

PDF, 124 KB

english, 1999

26

Condensed Heteroaromatic Ring Systems. XXIII. A Concise Synthesis of Hippadine

Sakamoto, Takao, Yasuhara, Akito, Kondo, Yoshinori, Yamanaka, Hiroshi

Journal:

Year:

1993

Language:

english

File:

PDF, 81 KB

english, 1993

27

MGS0039: a potent and selective group II metabotropic glutamate receptor antagonist with antidepressant-like activity

Shigeyuki Chaki, Ryoko Yoshikawa, Shiho Hirota, Toshiharu Shimazaki, Maoko Maeda, Naoya Kawashima, Takao Yoshimizu, Akito Yasuhara, Kazunari Sakagami, Shigeru Okuyama, Shigetada Nakanishi, Atsuro Naka

Journal:

Neuropharmacology

Year:

2004

Language:

english

File:

PDF, 381 KB

english, 2004

28

Synthesis, in Vitro Pharmacology, Structure−Activity Relationships, and Pharmacokinetics of 3-Alkoxy-2-amino-6-fluorobicyclo[3.1.0]hexane-2,6-dicarboxylic Acid Derivatives as Potent and Selective Group II Metabotropic Glutamate Receptor Antagonists

Nakazato, Atsuro, Sakagami, Kazunari, Yasuhara, Akito, Ohta, Hiroshi, Yoshikawa, Ryoko, Itoh, Manabu, Nakamura, Masato, Chaki, Shigeyuki

Journal:

Journal of Medicinal Chemistry

Year:

2004

Language:

english

File:

PDF, 215 KB

english, 2004

29

A Concise Synthesis of Furostifoline by Tetrabutylammonium Fluoride-Promoted Indole Ring Formation

Yasuhara, Akito, Suzuki, Naoyuki, Sakamoto, Takao

Journal:

CHEMICAL & PHARMACEUTICAL BULLETIN

Year:

2002

Language:

english

File:

PDF, 55 KB

english, 2002

30

Neuropharmacological profiles of antagonists of group II metabotropic glutamate receptors

Naoya Kawashima, Jun-ichi Karasawa, Toshiharu Shimazaki, Shigeyuki Chaki, Shigeru Okuyama, Akito Yasuhara, Atsuro Nakazato

Journal:

Neuroscience Letters

Year:

2005

Language:

english

File:

PDF, 103 KB

english, 2005

31

Deprotection of N-sulfonyl nitrogen-heteroaromatics with tetrabutylammonium fluoride

Akito Yasuhara, Takao Sakamoto

Journal:

Tetrahedron Letters

Year:

1998

Language:

english

File:

PDF, 90 KB

english, 1998

32

Condensed Heteroaromatic Ring Systems. XX. Palladium-Catalyzed Carbonylative Coupling of Iodobenzenes with (Z)-1-Ethoxy-2-(tributylstannyl)ethene.

SAKAMOTO, Takao, YASUHARA, Akito, KONDO, Yoshinori, YAMANAKA, Hiroshi

Journal:

CHEMICAL & PHARMACEUTICAL BULLETIN

Year:

1992

File:

PDF, 559 KB

1992

33

ChemInform Abstract: Selective Monodesulfonylation of N,N-Disulfonylarylamines with Tetrabutylammonium Fluoride.

Akito Yasuhara, Mitsuyoshi Kameda, Takao Sakamoto

Journal:

Year:

1999

File:

PDF, 32 KB

1999

34

ChemInform Abstract: Convenient Indole Synthesis from Ethynylanilines with a Polymer-Supported Fluoride.

Akito Yasuhara, Naoyuki Suzuki, Takashi Yoshino, Yousuke Takeda, Takao Sakamoto

Journal:

Year:

2002

File:

PDF, 28 KB

2002

35

ChemInform Abstract: Cyclization Reactions of 2-Alkynylbenzyl Alcohol and 2-Alkynylbenzylamine Derivatives Promoted by Tetrabutylammonium Fluoride.

Kou Hiroya, Rumi Jouka, Mitsuyoshi Kameda, Akito Yasuhara, Takao Sakamoto

Journal:

Year:

2002

File:

PDF, 33 KB

2002

36

Convenient Indole Synthesis from 2-Iodoanilines and Terminal Alkynes by the Sequential Sonogashira Reaction and the Cyclization Reaction Promoted by Tetrabutylammonium Fluoride (TBAF).

Naoyuki Suzuki, Sakura Yasaki, Akito Yasuhara, Takao Sakamoto

Journal:

Year:

2004

File:

PDF, 103 KB

2004

37

Convenient Indole Synthesis from 2-Iodoanilines and Terminal Alkynes by the Sequential Sonogashira Reaction and the Cyclization Reaction Promoted by Tetrabutylammonium Fluoride (TBAF)

Suzuki, Naoyuki, Yasaki, Sakura, Yasuhara, Akito, Sakamoto, Takao

Journal:

CHEMICAL & PHARMACEUTICAL BULLETIN

Year:

2003

Language:

english

File:

PDF, 59 KB

english, 2003

38

Synthesis of 2,3-Disubstituted Indole Using Palladium(II)-Catalyzed Cyclization with Alkenylation Reaction

Yasuhara, Akito, Takeda, Yousuke, Suzuki, Naoyuki, Sakamoto, Takao

Journal:

CHEMICAL & PHARMACEUTICAL BULLETIN

Year:

2002

Language:

english

File:

PDF, 63 KB

english, 2002

39

Synthesis, in vitro pharmacology, and pharmacokinetic profiles of 2-[1-amino-1-carboxy-2-(9H-xanthen-9-yl)-ethyl]-1-fluorocyclopropanecarboxylic acid and its 6-heptyl ester, a potent mGluR2 antagonist

Kazunari Sakagami, Akito Yasuhara, Shigeyuki Chaki, Ryoko Yoshikawa, Yasunori Kawakita, Akio Saito, Takeo Taguchi, Atsuro Nakazato

Journal:

Bioorganic & Medicinal Chemistry

Year:

2008

Language:

english

File:

PDF, 389 KB

english, 2008

40

ChemInform Abstract: Novel Synthetic Strategy of Carbolines via Palladium-Catalyzed Amination and Arylation Reaction.

Takehiko Iwaki, Akito Yasuhara, Takao Sakamoto

Journal:

Year:

1999

File:

PDF, 29 KB

1999

41

Prodrugs of 3-(3,4-dichlorobenzyloxy)-2-amino-6-fluorobicyclo[3.1.0]hexane-2,6-dicarboxylic acid (MGS0039): A potent and orally active group II mGluR antagonist with antidepressant-like potential

Akito Yasuhara, Masato Nakamura, Kazunari Sakagami, Toshiharu Shimazaki, Ryoko Yoshikawa, Shigeyuki Chaki, Hiroshi Ohta, Atsuro Nakazato

Journal:

Bioorganic & Medicinal Chemistry

Year:

2006

Language:

english

File:

PDF, 279 KB

english, 2006

To build up a library is to create a life. It’s never just a random collection of books.

— Carlos María Domínguez

Official channel

Z-Library Desktop Launcher

Z-Library Since 2009 support@1delivery.pm

EnglishРусскийEspañolItalianoελληνικάاللغة العربيةBahasa IndonesiaBahasa Malaysiaहिन्दीDeutschFrançaisPortuguêsУкраїнськаPolski中文繁體中文日本語Tiếng ViệtAzərbaycan DiliՀայոց լեզուภาษาไทยTürk Diliქართველიবাংলাپښتوతెలుగుاردو한국어SrpskiБългарски